Tamoxifen

Tamoxifen Citrate represent Selective estrogen receptor modulator (SERM).This drug is Widely used in medicine world as a treatment against breast cancer.Instead of the fact that Tamoxifen Citrate is a SERM, bodybuilders take it also as an anti-estrogen and as a triphenylethylene.Selective estrogen receptor modulators act as either estrogen receptor agonists or antagonists in a tissue-selective manner. The main reason why it is used by sportsmen, is the fact that it help to Prevent gynecomastia. Tamoxifen Citrate does this by competing for the receptor site in breast tissue, and binding to it. That's mean that act as tamoxifen and estrogen receptor blockade of breast tissue.Those bodybuilders / athletes who take Tamoxifen Citrate as a anti-estrogen supplement must remember that it is not the most efficient ancillary compound, but it is considering to be the safes. Tamoxifen Citrate does not actually reduce estrogen in human body, rather it blocks estrogen from estrogen receptors and, in those tissues where it is an antagonist, causes the receptor to do nothing.The usage of Tamoxifen Citrate has positive effects on immune system functionality as well as on lipid profile, on both HDL and LDL.Tamoxifen Citrate is chosen Often in post cycle therapy. After taking this drug hypogonadic and infertile men saw significant increase in the serum levels of LH, FSH, and testosterone levels as well. In fact, 20mgs of Tamoxifen can possibly raise testosterone levels approximately 150%Female bodybuilders / athletes usually take Tamoxifen Citrate in order to reduce the effect of endogenous estrogens Their Own. This can lower body fat concentrations, Especially in stubborn areas like the hips and thighs.Side effects that can occur are: in females - hot flashes, menstrual Irregularities and a variety of complications with the reproductive system, in males - reduced gains.
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Tamoxifen is an antagonist of the estrogen receptor in breast tissue via its active metabolite. The precise mechanism of its action is unknown, but one possibility is that it binds and blocks estrogen receptors on the surface of cells, preventing estrogens from binding and activating the cell.
40.00€
Nolvadex (Nolvadex)

Buy Nolvadex – Tamoxifen as an anti-estrogen (selective estrogen receptor modulator – SERM)

Brand name: Nolvadex (Tamoxifen Citrate)
Generic name: (Z)-2-[4-(1,2-diphenylbut-1-enyl)phenoxy]-N,N-dimethylethanamine
Producer / Manufacturer: Spectrum-Pharm

Tamoxifen is a drug called an estrogen receptor antagonist, which works by blocking the receptor so that estrogen can’t work its usual effects within the body.

Tamoxifen is an antagonist of the estrogen receptor in breast tissue via its active metabolite. The precise mechanism of its action is unknown, but one possibility is that it binds and blocks estrogen receptors on the surface of cells, preventing estrogens from binding and activating the cell. It is used in patients for treating and preventing breast cancer. Tamoxifen was approved by the FDA in December 1997.

Tamoxifen is used for the treatment of invasive breast cancer in men and women, the most common type of breast cancer, following surgery and/or radiation and for preventing invasive breast cancer in women at high risk for developing it. Tamoxifen also is used for the treatment of women following surgery and radiation for a less common type of breast cancer called ductal carcinoma in situ (DCIS or intraductal carcinoma). Women who have had DCIS are at high risk for developing invasive breast cancer at a later date, and tamoxifen prevents development of the invasive cancer in almost half of the women during the first five years of treatment. Occasionally, tamoxifen is used to stimulate ovulation.

Estrogen is an important hormone in the female body and plays a big role in some types of breast cancer. As a result, tamoxifen is commonly used to prevent breast cancer from appearing or coming back in women who are at a high risk of or have a history of breast cancer.
This is not the only way that tamoxifen can be used, however, and there are several alternative ways that this drug can be used to offer a benefit. The following information goes into more detail about alternative uses of the medication and how it can be used.

Tamoxifen Citrate has been used medically for decades and has been highly successful in breast cancer treatment, specifically hormone-responsive breast cancer. It is also a medication that is used by many anabolic steroid users, but it is not a steroid. This is a drug steroid users will sometimes use during steroid use to help with estrogenic related side effects brought on by specific steroids. However, it is most commonly used during Post Cycle Therapy (PCT). PCT is the 3-6 week period following steroid use that is implemented in order to help with natural testosterone production that is suppressed during anabolic steroid use.

Tamoxifen Citrate Functions & Traits

Tamoxifen Citrate is a SERM that acts as both antagonist and agonist in relation to the estrogen hormone. It is an anti-estrogen in that it binds to estrogen receptors in certain parts of the body, particularly in the mammary tissue. This action prevents estrogen from acting on its originally intended point of binding. This makes Tamoxifen Citrate valuable to breast cancer patients as breast cancer feeds off of estrogen. And it’s valuable to steroid users as increased estrogen levels can bind to the mammary tissue and lead to gynecomastia.

The relationship Tamoxifen Citrate has in being an anti-estrogen is fairly straightforward and well understood by many, but it’s its relationship to being an estrogen in other areas that’s surprising to some. Tamoxifen Citrate acts as an estrogen on the liver. Liver related estrogenic activity has been shown to improve cardiovascular health, particularly as it relates to cholesterol. This can be very advantageous for the bodybuilding steroid user as most steroids have a negative impact on cholesterol levels.

Beyond its estrogen related activity Tamoxifen Citrate possesses strong testosterone stimulating properties. The use of Tamoxifen Citrate will stimulate the pituitary to increase its production of Luteinizing Hormone (LH) and Follicle Stimulating Hormone (FSH) with a strong emphasis on LH. LH and FSH are the gonadotropins that signal to the testicles to produce testosterone.

Effects of Tamoxifen Citrate

For the anabolic steroid user the positive effects of Tamoxifen Citrate can be seen both during and post anabolic steroid use with post use being primary. Anabolic steroids like Testosterone and Nandrolone among others will increase the body’s serum estrogen levels. This occurs by the testosterone hormone converting to testosterone, which happens due to it being metabolized by the aromatase enzyme. Once aromatized you have more estrogen, and this can lead to gynecomastia and water retention. It can also lead to high blood pressure if water retention becomes severe. Tamoxifen Citrate does not lower serum estrogen levels, but it will bind to the receptors in the chest preventing the estrogen from binding. It will not do a lot for water retention if that is an issue. It is also not enough gynecomastia protection for all men, but that depends on how high estrogen levels go as well as genetics. If more or stronger protection is needed Aromatase Inhibitors (AI’s) are recommended. AI’s are anti-estrogens that inhibit aromatase activity and lower serum estrogen levels.

We then have the testosterone stimulating effects of Tamoxifen Citrate. This is by far the most important effect for the anabolic steroid user. When we use anabolic steroids we suppress our natural testosterone production, and this will occur regardless of the steroids used. Steroid use creates a negative feedback and tells your pituitary to stop making LH and FSH. This is why almost all steroid cycles include exogenous testosterone so that the negative feedback doesn’t cause a low testosterone level. Once steroid use is complete something is then needed to jump start testosterone production. It will occur on its own, but it will be slow and Tamoxifen can both speed it up and make it more efficient. Tamoxifen Citrate is introduced, LH and FSH levels go up and as a result testosterone is produced.

Important Note: PCT use that includes Tamoxifen Citrate or any SERM, for it to be successful this assumes no prior low testosterone condition existed. It also assumes no damage was done to the Hypothalamic-Pituitary-Testicular-Axis (HPTA) during use. If prior low levels existed Tamoxifen Citrate won’t magically fix this. If severe damage was done to the HPTA you will not recover and may be in need of low testosterone treatment.

Important Note: Many steroid users believe that a good PCT brings about full recovery, but this is a false belief. A PCT that includes Tamoxifen Citrate will stimulate recovery, but it will not end it. It will still take several months for full recovery to occur, but it stands a much better chance with PCT than without.

Anabolic steroids trade names:

Stubal
Valodex
Genox
Adifen
Soltamox
Adopan
Bagotam
Bilem
Bioxifeno
Citofen
Crisafeno
Doctamoxifene
Ebefen
Istubal
Valodex
Genox
Emalook
Femoxtal
Fenobest
Ginarsan
Gynatam
Mamofen
Neophedan
Nolgen
Nomafen
Norxifen
Novofen
Oncotamox
Panleef
Phenolurn
Puretam
Respol
Rolap
Tamec
Tamifen
Tamizam
Tamokadin
Tamona
Tamoneprin
Tamophar
Tamosin
Tamoxen
Tamoxene
Tamoxi
Tamoxifène
Tamoxin
Tamoxis
Tamoxistad
Tamsulon
Tasuomin
Taxfeno
Tecnotax
Trimetrox
Yacesal
Zymoplex



COMMON
Active substanceTamoxifen citrate
IndicationsBlocks estrogen & prevents gynecomastia. Increases natural testosterone levels.
DOSAGE
Quantity25-75
UnitMilligram
TimeDay
POTENCY
Quantity25
UnitMilligram/Tablet
PACKAGING
Quantity100
UnitTablet
TypePlastic bottle
Presentation100 tablets, packed & sealed in white HDPE plastic bottle.
Tamoxifen is an antagonist of the estrogen receptor in breast tissue via its active metabolite. The precise mechanism of its action is unknown, but one possibility is that it binds and blocks estrogen receptors on the surface of cells, preventing estrogens from binding and activating the cell.
40.00€
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